Strategic Use of Benzylic Alcohols Reveals Cryptic Hydrogen-Bonding Interactions: Discovery of HBC-12551 as a Potent Noncovalent Bruton's Tyrosine Kinase Inhibitor. uri icon

authors

  • Liu, Gang
  • Zhu, Hugh
  • Chang, Tzu-Pei
  • Max, Nathan
  • Manish Kumar, MD
  • Chen, Cynthia
  • Lee, Lance
  • Liu, Shuaishuai
  • Cho, Sangwoo
  • Chae, Hee-Don
  • Zhou, Wei
  • Zhang, Lingtian
  • Khanna, Avinash
  • Zeng, Xin
  • Du, Xinlin

publication date

  • January 30, 2026